Assay Detail
Binding
CHEMBL5152645
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Competitive inhibition of recombinant human MAO-B using kynuramine as substrate assessed as enzyme-inhibitor dissociation constant at varying substrate concentration by Lineweaver-burk plot analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
The inhibition of monoamine oxidase by 2H-1,4-benzothiazin-3(4H)-ones.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 8.17 | 8.17 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5174014 | — | — | 1 | 8.17 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5174014 | — | Ki | = | 6.7 | nM | 8.17 |