Assay Detail
Binding
CHEMBL5153459
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Binding affinity to BCL6 (unknown origin) by TR-FRET assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
B-cell Lymphoma 6 Inhibitors: Current Advances and Prospects of Drug Development for Diffuse Large B-cell Lymphomas.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 7.49 | 8.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5184651 | — | — | 1 | 8.05 |
| CHEMBL5207356 | — | — | 1 | 6.92 |
| CHEMBL1721570 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5184651 | — | IC50 | = | 8.9 | nM | 8.05 |
| CHEMBL5207356 | — | IC50 | = | 120.0 | nM | 6.92 |
| CHEMBL1721570 | — | IC50 | = | 830000.0 | nM | - |