Assay Detail
Functional
CHEMBL5158256
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assay
49
Total Activities
48
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CHO-RD-HGA16 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Neuropeptides B/W receptor type 1 (CHEMBL1293293) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Neuropeptide B/W receptor 1 peptidomimetic agonists: Structure-activity relationships and plasma stability.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 48 | 7.20 | 8.10 |
| EC80 | 1 | - | - |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5187335 | — | — | 1 | 8.10 |
| CHEMBL5170622 | — | — | 2 | 8.10 |
| CHEMBL5194519 | — | — | 1 | 7.96 |
| CHEMBL5178929 | — | — | 1 | 7.96 |
| CHEMBL5172042 | — | — | 1 | 7.89 |
| CHEMBL5206425 | — | — | 1 | 7.89 |
| CHEMBL5177662 | — | — | 1 | 7.85 |
| CHEMBL5188323 | — | — | 1 | 7.70 |
| CHEMBL5179908 | — | — | 1 | 7.66 |
| CHEMBL5191528 | — | — | 1 | 7.66 |
| CHEMBL5204006 | — | — | 1 | 7.64 |
| CHEMBL5197385 | — | — | 1 | 7.60 |
| CHEMBL5208352 | — | — | 1 | 7.39 |
| CHEMBL5174290 | — | — | 1 | 7.32 |
| CHEMBL5189212 | — | — | 1 | 7.24 |
| CHEMBL5195844 | — | — | 1 | 7.23 |
| CHEMBL5194208 | — | — | 1 | 7.20 |
| CHEMBL5185639 | — | — | 1 | 7.03 |
| CHEMBL5200286 | — | — | 1 | 7.01 |
| CHEMBL5191389 | — | — | 1 | 6.95 |
| CHEMBL5180015 | — | — | 1 | 6.71 |
| CHEMBL5190117 | — | — | 1 | 6.65 |
| CHEMBL5180153 | — | — | 1 | 6.39 |
| CHEMBL5182424 | — | — | 1 | 6.33 |
| CHEMBL5197610 | — | — | 1 | 6.32 |
| CHEMBL5185495 | — | — | 1 | 6.32 |
| CHEMBL5198287 | — | — | 1 | 6.28 |
| CHEMBL5203099 | — | — | 1 | 6.24 |
| CHEMBL5202376 | — | — | 1 | 6.12 |
| CHEMBL5186704 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5187335 | — | EC50 | = | 8.0 | nM | 8.10 |
| CHEMBL5170622 | — | EC50 | = | 8.0 | nM | 8.10 |
| CHEMBL5178929 | — | EC50 | = | 11.0 | nM | 7.96 |
| CHEMBL5194519 | — | EC50 | = | 10.9 | nM | 7.96 |
| CHEMBL5172042 | — | EC50 | = | 13.0 | nM | 7.89 |
| CHEMBL5206425 | — | EC50 | = | 13.0 | nM | 7.89 |
| CHEMBL5177662 | — | EC50 | = | 14.0 | nM | 7.85 |
| CHEMBL5188323 | — | EC50 | = | 20.0 | nM | 7.70 |
| CHEMBL5179908 | — | EC50 | = | 22.0 | nM | 7.66 |
| CHEMBL5191528 | — | EC50 | = | 22.0 | nM | 7.66 |
| CHEMBL5204006 | — | EC50 | = | 23.0 | nM | 7.64 |
| CHEMBL5197385 | — | EC50 | = | 25.0 | nM | 7.60 |
| CHEMBL5208352 | — | EC50 | = | 41.0 | nM | 7.39 |
| CHEMBL5174290 | — | EC50 | = | 48.0 | nM | 7.32 |
| CHEMBL5189212 | — | EC50 | = | 57.0 | nM | 7.24 |
| CHEMBL5195844 | — | EC50 | = | 59.0 | nM | 7.23 |
| CHEMBL5194208 | — | EC50 | = | 63.0 | nM | 7.20 |
| CHEMBL5185639 | — | EC50 | = | 93.0 | nM | 7.03 |
| CHEMBL5200286 | — | EC50 | = | 98.0 | nM | 7.01 |
| CHEMBL5191389 | — | EC50 | = | 112.0 | nM | 6.95 |
| CHEMBL5180015 | — | EC50 | = | 194.0 | nM | 6.71 |
| CHEMBL5190117 | — | EC50 | = | 225.0 | nM | 6.65 |
| CHEMBL5180153 | — | EC50 | = | 406.0 | nM | 6.39 |
| CHEMBL5182424 | — | EC50 | = | 463.0 | nM | 6.33 |
| CHEMBL5185495 | — | EC50 | = | 479.0 | nM | 6.32 |
| CHEMBL5197610 | — | EC50 | = | 478.0 | nM | 6.32 |
| CHEMBL5198287 | — | EC50 | = | 530.0 | nM | 6.28 |
| CHEMBL5203099 | — | EC50 | = | 578.0 | nM | 6.24 |
| CHEMBL5202376 | — | EC50 | = | 766.0 | nM | 6.12 |
| CHEMBL5186704 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5199142 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5200724 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5183635 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5174076 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5190871 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5171882 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5170866 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5186461 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5175824 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5196275 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5194363 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5195516 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5198182 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5170622 | — | EC80 | = | 20.0 | nM | - |
| CHEMBL5178251 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5202561 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5180498 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5188509 | — | EC50 | > | 10000.0 | nM | - |
| CHEMBL5177589 | — | EC50 | > | 10000.0 | nM | - |