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Assay Detail

CHEMBL5159787

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Binding
Binding affinity to influenza A virus RNA-dependent RNA polymerase PB1 subunit expressed in human 293T cells assessed as dissociation constant by MST assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Influenza A virus
Cell Type HEK293T
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Discovery of Aryl Benzoyl Hydrazide Derivatives as Novel Potent Broad-Spectrum Inhibitors of Influenza A Virus RNA-Dependent RNA Polymerase (RdRp).
Liu X, Liang J, Yu Y, Han X, Yu L, Chen F, Xu Z, Chen Q, Jin M, Dong C, Zhou HB, Lan K, Wu S.
J Med Chem (2022) 65 : 3814 -3832
PubMed 35212527 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 1 6.46 6.46

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5194584 1 6.46

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5194584 Kd = 351.0 nM 6.46