Assay Detail
Functional
CHEMBL5161545
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antirabies activity against rabies CVS infected in golden hamster BSR cells preincubated for 1 hr followed by mixing of cells measured after 24 hrs by inverted fluorescence microscope analysis
33
Total Activities
33
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Lyssavirus rabies |
| Cell Type | BSR |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Clofazimine derivatives as potent broad-spectrum antiviral agents with dual-target mechanism.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 33 | 5.32 | 6.12 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5172292 | — | — | 1 | 6.12 |
| CHEMBL351554 | — | — | 1 | 6.12 |
| CHEMBL5200072 | — | — | 1 | 5.85 |
| CHEMBL5187097 | — | — | 1 | 5.85 |
| CHEMBL5206254 | — | — | 1 | 5.85 |
| CHEMBL5183417 | — | — | 1 | 5.84 |
| CHEMBL5183802 | — | — | 1 | 5.78 |
| CHEMBL5192145 | — | — | 1 | 5.75 |
| CHEMBL5181774 | — | — | 1 | 5.72 |
| CHEMBL5202017 | — | — | 1 | 5.72 |
| CHEMBL1292 | CLOFAZIMINE | 4.0 | 1 | 5.64 |
| CHEMBL5189682 | — | — | 1 | 5.64 |
| CHEMBL5182140 | — | — | 1 | 5.64 |
| CHEMBL5172591 | — | — | 1 | 5.59 |
| CHEMBL5189244 | — | — | 1 | 5.40 |
| CHEMBL5184086 | — | — | 1 | 5.34 |
| CHEMBL5171443 | — | — | 1 | 5.30 |
| CHEMBL5203269 | — | — | 1 | 5.30 |
| CHEMBL5190503 | — | — | 1 | 5.16 |
| CHEMBL5201337 | — | — | 1 | 5.16 |
| CHEMBL5180232 | — | — | 1 | 5.16 |
| CHEMBL5178249 | — | — | 1 | 5.07 |
| CHEMBL152430 | — | — | 1 | 4.97 |
| CHEMBL5186686 | — | — | 1 | 4.91 |
| CHEMBL5181861 | — | — | 1 | 4.88 |
| CHEMBL5173971 | — | — | 1 | 4.88 |
| CHEMBL5174821 | — | — | 1 | 4.69 |
| CHEMBL358684 | — | — | 1 | 4.69 |
| CHEMBL5171985 | — | — | 1 | 4.64 |
| CHEMBL422348 | — | — | 1 | 4.60 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5172292 | — | EC50 | = | 760.0 | nM | 6.12 |
| CHEMBL351554 | — | EC50 | = | 760.0 | nM | 6.12 |
| CHEMBL5200072 | — | EC50 | = | 1400.0 | nM | 5.85 |
| CHEMBL5187097 | — | EC50 | = | 1410.0 | nM | 5.85 |
| CHEMBL5206254 | — | EC50 | = | 1400.0 | nM | 5.85 |
| CHEMBL5183417 | — | EC50 | = | 1450.0 | nM | 5.84 |
| CHEMBL5183802 | — | EC50 | = | 1670.0 | nM | 5.78 |
| CHEMBL5192145 | — | EC50 | = | 1770.0 | nM | 5.75 |
| CHEMBL5181774 | — | EC50 | = | 1900.0 | nM | 5.72 |
| CHEMBL5202017 | — | EC50 | = | 1900.0 | nM | 5.72 |
| CHEMBL1292 | CLOFAZIMINE | EC50 | = | 2280.0 | nM | 5.64 |
| CHEMBL5189682 | — | EC50 | = | 2290.0 | nM | 5.64 |
| CHEMBL5182140 | — | EC50 | = | 2290.0 | nM | 5.64 |
| CHEMBL5172591 | — | EC50 | = | 2550.0 | nM | 5.59 |
| CHEMBL5189244 | — | EC50 | = | 4020.0 | nM | 5.40 |
| CHEMBL5184086 | — | EC50 | = | 4560.0 | nM | 5.34 |
| CHEMBL5171443 | — | EC50 | = | 5030.0 | nM | 5.30 |
| CHEMBL5203269 | — | EC50 | = | 5030.0 | nM | 5.30 |
| CHEMBL5190503 | — | EC50 | = | 6860.0 | nM | 5.16 |
| CHEMBL5201337 | — | EC50 | = | 6860.0 | nM | 5.16 |
| CHEMBL5180232 | — | EC50 | = | 6860.0 | nM | 5.16 |
| CHEMBL5178249 | — | EC50 | = | 8440.0 | nM | 5.07 |
| CHEMBL152430 | — | EC50 | = | 10700.0 | nM | 4.97 |
| CHEMBL5186686 | — | EC50 | = | 12300.0 | nM | 4.91 |
| CHEMBL5181861 | — | EC50 | = | 13200.0 | nM | 4.88 |
| CHEMBL5173971 | — | EC50 | = | 13200.0 | nM | 4.88 |
| CHEMBL5174821 | — | EC50 | = | 20600.0 | nM | 4.69 |
| CHEMBL358684 | — | EC50 | = | 20600.0 | nM | 4.69 |
| CHEMBL5171985 | — | EC50 | = | 22700.0 | nM | 4.64 |
| CHEMBL422348 | — | EC50 | = | 24900.0 | nM | 4.60 |
| CHEMBL5180416 | — | EC50 | = | 35400.0 | nM | 4.45 |
| CHEMBL5205379 | — | EC50 | = | 35400.0 | nM | 4.45 |
| CHEMBL5182002 | — | EC50 | = | 106000.0 | nM | - |