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Assay Detail

CHEMBL5163707

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of deltaC55 truncated Hepatitis C virus NS5B expressed in Escherichia coli using poly(rA)/oligo(rU) as template/primer incubated for 20 mins in presence of 3H-UTP by radioactivity based assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Hepatitis C virus
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

RNA-directed RNA polymerase (CHEMBL4296320)
Type SINGLE PROTEIN
Organism Hepacivirus hominis

Publication

4,5-Dihydroxypyrimidine Methyl Carboxylates, Carboxylic Acids, and Carboxamides as Inhibitors of Human Cytomegalovirus pUL89 Endonuclease.
He T, Edwards TC, Xie J, Aihara H, Geraghty RJ, Wang Z.
J Med Chem (2022) 65 : 5830 -5849
PubMed 35377638 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.58 5.58

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL181653 1 5.58

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL181653 IC50 = 2600.0 nM 5.58