Assay Detail
Binding
CHEMBL5209673
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Cellular target engagement assay with: FGFR2
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | HEK-293T |
| Category | NanoBRET assay |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
NanoBRET assay results for EUbOPEN Chemogenomics Library 3
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 7.60 | 7.60 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL189584 | PD-173074 | — | 1 | 7.60 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL189584 | PD-173074 | IC50 | = | 25.1 | nM | 7.60 |