Assay Detail

CHEMBL5213261

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Binding

Selectivity interaction (Enzymatic assay) EUB0000305b STK17A

ChEMBL ↗

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Target

Serine/threonine-protein kinase 17A (CHEMBL4525) ↗

Open DB target context

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Serine/threonine-protein kinase 17A (CHEMBL4525) is the working anchor for this assay review. Loading the live Open DB target snapshot…

Primary target Serine/threonine-protein kinase 17A

CHEMBL4525

Anchored from Assay target.

Protein identity Serine/threonine-protein kinase 17A

Disease frame Disease evidence pending

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Review focus Open DB context pending

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Total Activities

Compounds Tested

Activity Types

Assay Parameters

Assay Information

Assay Type	Binding
Organism	Homo sapiens
Category	Selectivity assay
Confidence	9 — Direct single protein target
Curated By	Autocuration

Target

Serine/threonine-protein kinase 17A (CHEMBL4525) ↗

Type	SINGLE PROTEIN
Organism	Homo sapiens

Publication

Selectivity Literature for EUbOPEN Chemogenomics Library wave 3

EUbOPEN
(2023)
· DOI

Activity Statistics

Type	Count	Avg pChEMBL	Best pChEMBL
IC50	1	6.51	6.51

Assay Parameters

Parameter	Type	Value	Units	Text
Protein family	Protein family	-	—	Protein Kinase

Compounds Tested

Compound	Name	Phase	Activities	Best pChEMBL
CHEMBL4537673	BAY-985	—	1	6.51

Activity Data

Compound	Name	Type	Rel.	Value	Units	pChEMBL
CHEMBL4537673	BAY-985	IC50	=	311.0	nM	6.51