Assay Detail
Binding
CHEMBL5216041
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of MCT1 in rat erythrocytes
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Cell Type | Erythrocyte |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Monocarboxylate transporter 1 (CHEMBL2073709) ↗| Type | SINGLE PROTEIN |
| Organism | Rattus norvegicus |
Publication
Novel strategies to improve tumour therapy by targeting the proteins MCT1, MCT4 and LAT1.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 8.64 | 8.64 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5221129 | — | — | 1 | 8.64 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5221129 | — | Ki | = | 2.3 | nM | 8.64 |