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Assay Detail

CHEMBL5216355

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antibacterial activity against Bacillus subtilis NCIM 2079 assessed as reduction in bacterial growth incubated for 8 hrs by absorbance based assay
9
Total Activities
9
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Bacillus subtilis
Confidence 1 — Organism
Curated By Autocuration

Target

Bacillus subtilis (CHEMBL359)
Type ORGANISM
Organism Bacillus subtilis

Publication

Recent contribution of medicinally active 2-aminothiophenes: A privileged scaffold for drug discovery.
Duvauchelle V, Meffre P, Benfodda Z.
Eur J Med Chem (2022) 238 : 114502 -114502
PubMed 35696863 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 9 6.68 6.82

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5218479 1 6.82
CHEMBL174 AMPICILLIN 4.0 1 6.82
CHEMBL1082 AMOXICILLIN 4.0 1 6.82
CHEMBL5219555 1 6.68
CHEMBL5220084 1 6.68
CHEMBL5219187 1 6.60
CHEMBL1727 CEPHALEXIN ANHYDROUS 4.0 1 6.60
CHEMBL5219360 1 6.58
CHEMBL5220992 1 6.55

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5218479 EC50 = 150.0 nM 6.82
CHEMBL174 AMPICILLIN EC50 = 150.0 nM 6.82
CHEMBL1082 AMOXICILLIN EC50 = 150.0 nM 6.82
CHEMBL5219555 EC50 = 210.0 nM 6.68
CHEMBL5220084 EC50 = 210.0 nM 6.68
CHEMBL5219187 EC50 = 250.0 nM 6.60
CHEMBL1727 CEPHALEXIN ANHYDROUS EC50 = 250.0 nM 6.60
CHEMBL5219360 EC50 = 260.0 nM 6.58
CHEMBL5220992 EC50 = 280.0 nM 6.55