Assay Detail
Binding
CHEMBL5216513
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Inhibition of human IDO1
24
Total Activities
24
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery of the First Selective IDO2 Inhibitor As Novel Immunotherapeutic Avenues for Rheumatoid Arthritis.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 24 | 7.20 | 7.55 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5091825 | — | — | 1 | 7.55 |
| CHEMBL5221037 | — | — | 1 | 7.43 |
| CHEMBL5220224 | — | — | 1 | 7.33 |
| CHEMBL5221035 | — | — | 1 | 7.28 |
| CHEMBL5219888 | — | — | 1 | 6.39 |
| CHEMBL5219050 | — | — | 1 | - |
| CHEMBL5219670 | — | — | 1 | - |
| CHEMBL5219166 | — | — | 1 | - |
| CHEMBL5221052 | — | — | 1 | - |
| CHEMBL5219627 | — | — | 1 | - |
| CHEMBL5220174 | — | — | 1 | - |
| CHEMBL5220058 | — | — | 1 | - |
| CHEMBL5220112 | — | — | 1 | - |
| CHEMBL5219521 | — | — | 1 | - |
| CHEMBL5218706 | — | — | 1 | - |
| CHEMBL5220905 | — | — | 1 | - |
| CHEMBL5218638 | — | — | 1 | - |
| CHEMBL5220365 | — | — | 1 | - |
| CHEMBL5218514 | — | — | 1 | - |
| CHEMBL5219143 | — | — | 1 | - |
| CHEMBL5218855 | — | — | 1 | - |
| CHEMBL5218715 | — | — | 1 | - |
| CHEMBL5219677 | — | — | 1 | - |
| CHEMBL5220617 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5091825 | — | IC50 | = | 28.0 | nM | 7.55 |
| CHEMBL5221037 | — | IC50 | = | 37.0 | nM | 7.43 |
| CHEMBL5220224 | — | IC50 | = | 47.0 | nM | 7.33 |
| CHEMBL5221035 | — | IC50 | = | 52.0 | nM | 7.28 |
| CHEMBL5219888 | — | IC50 | = | 411.0 | nM | 6.39 |
| CHEMBL5219050 | — | IC50 | - | — | - | |
| CHEMBL5219670 | — | IC50 | - | — | - | |
| CHEMBL5219166 | — | IC50 | - | — | - | |
| CHEMBL5221052 | — | IC50 | - | — | - | |
| CHEMBL5219627 | — | IC50 | - | — | - | |
| CHEMBL5220174 | — | IC50 | - | — | - | |
| CHEMBL5220058 | — | IC50 | - | — | - | |
| CHEMBL5220112 | — | IC50 | - | — | - | |
| CHEMBL5219521 | — | IC50 | - | — | - | |
| CHEMBL5218706 | — | IC50 | - | — | - | |
| CHEMBL5220905 | — | IC50 | - | — | - | |
| CHEMBL5218638 | — | IC50 | - | — | - | |
| CHEMBL5220365 | — | IC50 | - | — | - | |
| CHEMBL5218514 | — | IC50 | - | — | - | |
| CHEMBL5219143 | — | IC50 | - | — | - | |
| CHEMBL5218855 | — | IC50 | - | — | - | |
| CHEMBL5218715 | — | IC50 | - | — | - | |
| CHEMBL5219677 | — | IC50 | - | — | - | |
| CHEMBL5220617 | — | IC50 | - | — | - |