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Assay Detail

CHEMBL5217630

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Binding
Inhibition of Keap1 kelch domain to Nrf2 (unknown origin) protein-protein interaction
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 5 — Multiple protein complex / RNA
Curated By Autocuration

Target

Keap1/Nrf2 (CHEMBL3038498)
Type PROTEIN-PROTEIN INTERACTION
Organism Homo sapiens

Publication

Development of Noncovalent Small-Molecule Keap1-Nrf2 Inhibitors by Fragment-Based Drug Discovery.
Narayanan D, Tran KT, Pallesen JS, Solbak SMØ, Qin Y, Mukminova E, Luchini M, Vasilyeva KO, González Chichón D, Goutsiou G, Poulsen C, Haapanen N, Popowicz GM, Sattler M, Olagnier D, Gajhede M, Bach A.
J Med Chem (2022) 65 : 14481 -14526
PubMed 36263945 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 6 7.16 7.66

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4739983 1 7.66
CHEMBL4174651 1 7.22
CHEMBL4646536 1 7.14
CHEMBL4740287 1 7.12
CHEMBL5219681 1 7.01
CHEMBL4640621 1 6.82

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4739983 IC50 = 22.0 nM 7.66
CHEMBL4174651 IC50 = 60.0 nM 7.22
CHEMBL4646536 IC50 = 73.0 nM 7.14
CHEMBL4740287 IC50 = 75.0 nM 7.12
CHEMBL5219681 IC50 = 97.0 nM 7.01
CHEMBL4640621 IC50 = 150.0 nM 6.82