Assay Detail
Binding
CHEMBL5218423
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to PPARdelta (unknown origin) assessed as inhibition constant by Cheng-Prusoff equation analysis
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Peroxisome proliferator-activated receptor delta (CHEMBL3979) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Discovery of Pan-peroxisome Proliferator-Activated Receptor Modulators from an Endolichenic Fungus, <i>Daldinia childiae</i>.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 6.87 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL38943 | GW501516 | 2.0 | 1 | 9.00 |
| CHEMBL5219536 | — | — | 1 | 4.73 |
| CHEMBL5220260 | — | — | 1 | - |
| CHEMBL595 | PIOGLITAZONE | 4.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL38943 | GW501516 | Ki | = | 1.0 | nM | 9.00 |
| CHEMBL5219536 | — | Ki | = | 18800.0 | nM | 4.73 |
| CHEMBL5220260 | — | Ki | - | — | - | |
| CHEMBL595 | PIOGLITAZONE | Ki | - | — | - |