Assay Detail
Binding
CHEMBL5223233
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antagonist activity at CXCR2 (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Recent advances in urea- and thiourea-containing compounds: focus on innovative approaches in medicinal chemistry and organic synthesis.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 8.65 | 8.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5276296 | — | — | 1 | 8.70 |
| CHEMBL216981 | NAVARIXIN ANHYDROUS | 2.0 | 1 | 8.59 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5276296 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL216981 | NAVARIXIN ANHYDROUS | IC50 | = | 2.6 | nM | 8.59 |