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Assay Detail

CHEMBL5223543

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Functional
Antiproliferative activity against human HT-29 cells assessed as cell growth inhibition
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type HT-29
Confidence 1 — Organism
Curated By Autocuration

Target

HT-29 (CHEMBL384)
Type CELL-LINE
Organism Homo sapiens

Publication

Recent advances on synthesis and biological activities of aurones.
Sui G, Li T, Zhang B, Wang R, Hao H, Zhou W.
Bioorg Med Chem (2021) 29 : 115895 -115895
PubMed 33271454 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 6 5.24 5.38

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL326574 1 5.38
CHEMBL326079 1 5.38
CHEMBL324265 1 5.37
CHEMBL113771 1 5.23
CHEMBL115120 1 5.05
CHEMBL116391 1 5.04

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL326574 IC50 = 4120.0 nM 5.38
CHEMBL326079 IC50 = 4120.0 nM 5.38
CHEMBL324265 IC50 = 4320.0 nM 5.37
CHEMBL113771 IC50 = 5900.0 nM 5.23
CHEMBL115120 IC50 = 8900.0 nM 5.05
CHEMBL116391 IC50 = 9120.0 nM 5.04