Assay Detail
Binding
CHEMBL5223601
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human BCL6 BTP domain measured by TR-FRET assay
16
Total Activities
16
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Progress toward B-Cell Lymphoma 6 BTB Domain Inhibitors for the Treatment of Diffuse Large B-Cell Lymphoma and Beyond.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 16 | 6.86 | 8.54 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4094351 | — | — | 1 | 8.54 |
| CHEMBL5184651 | — | — | 1 | 8.05 |
| CHEMBL4064865 | — | — | 1 | 7.96 |
| CHEMBL4092565 | — | — | 1 | 7.92 |
| CHEMBL4100303 | — | — | 1 | 7.89 |
| CHEMBL5277976 | — | — | 1 | 7.34 |
| CHEMBL5273385 | — | — | 1 | 7.20 |
| CHEMBL5207356 | — | — | 1 | 6.92 |
| CHEMBL4061857 | — | — | 1 | 6.46 |
| CHEMBL4077836 | — | — | 1 | 6.43 |
| CHEMBL4445645 | — | — | 1 | 6.28 |
| CHEMBL4547183 | — | — | 1 | 6.12 |
| CHEMBL4572689 | — | — | 1 | 6.07 |
| CHEMBL4542555 | — | — | 1 | 5.47 |
| CHEMBL4065661 | — | — | 1 | 4.21 |
| CHEMBL1721570 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4094351 | — | IC50 | = | 2.9 | nM | 8.54 |
| CHEMBL5184651 | — | IC50 | = | 8.9 | nM | 8.05 |
| CHEMBL4064865 | — | IC50 | = | 11.0 | nM | 7.96 |
| CHEMBL4092565 | — | IC50 | = | 12.0 | nM | 7.92 |
| CHEMBL4100303 | — | IC50 | = | 13.0 | nM | 7.89 |
| CHEMBL5277976 | — | IC50 | = | 46.0 | nM | 7.34 |
| CHEMBL5273385 | — | IC50 | = | 63.0 | nM | 7.20 |
| CHEMBL5207356 | — | IC50 | = | 120.0 | nM | 6.92 |
| CHEMBL4061857 | — | IC50 | = | 350.0 | nM | 6.46 |
| CHEMBL4077836 | — | IC50 | = | 370.0 | nM | 6.43 |
| CHEMBL4445645 | — | IC50 | = | 520.0 | nM | 6.28 |
| CHEMBL4547183 | — | IC50 | = | 760.0 | nM | 6.12 |
| CHEMBL4572689 | — | IC50 | = | 860.0 | nM | 6.07 |
| CHEMBL4542555 | — | IC50 | = | 3400.0 | nM | 5.47 |
| CHEMBL4065661 | — | IC50 | = | 61000.0 | nM | 4.21 |
| CHEMBL1721570 | — | IC50 | = | 830000.0 | nM | - |