Assay Detail
Binding
CHEMBL5223603
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Inhibition of CK2 (unknown origin)
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Publication
Progress toward B-Cell Lymphoma 6 BTB Domain Inhibitors for the Treatment of Diffuse Large B-Cell Lymphoma and Beyond.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 4 | 6.19 | 6.19 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4094351 | — | — | 1 | 6.19 |
| CHEMBL4100303 | — | — | 1 | - |
| CHEMBL4092565 | — | — | 1 | - |
| CHEMBL4064865 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4094351 | — | IC50 | = | 640.0 | nM | 6.19 |
| CHEMBL4100303 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4092565 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4064865 | — | IC50 | > | 10000.0 | nM | - |