Assay Detail
Binding
CHEMBL5223809
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of farnesyltransferase in human Burkitts lymphoma cell
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | Burkitts lymphoma cell |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Targeting Small GTPases and Their Prenylation in Diabetes Mellitus.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.73 | 8.85 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL431828 | — | — | 1 | 8.85 |
| CHEMBL1258350 | — | — | 1 | 6.60 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL431828 | — | IC50 | = | 1.4 | nM | 8.85 |
| CHEMBL1258350 | — | IC50 | = | 250.0 | nM | 6.60 |