Assay Detail
Binding
CHEMBL5224079
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to LSD1 (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Lysine-specific histone demethylase 1A (CHEMBL6136) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Annual review of lysine-specific demethylase 1 (LSD1/KDM1A) inhibitors in 2021.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 2 | 6.02 | 6.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5093633 | — | — | 1 | 6.62 |
| CHEMBL5075646 | — | — | 1 | 5.42 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5093633 | — | Kd | = | 240.0 | nM | 6.62 |
| CHEMBL5075646 | — | Kd | = | 3830.0 | nM | 5.42 |