Assay Detail
Binding
CHEMBL5225167
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Inhibition of human MMP2
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
A review of MMP-2 structures and binding mode analysis of its inhibitors to strategize structure-based drug design.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.64 | 7.57 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5283314 | — | — | 1 | 7.57 |
| CHEMBL460657 | ELAIDIC ACID | — | 1 | 5.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5283314 | — | IC50 | = | 27.0 | nM | 7.57 |
| CHEMBL460657 | ELAIDIC ACID | IC50 | = | 1995.0 | nM | 5.70 |