Assay Detail
Binding
CHEMBL5226441
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Inhibition of HDAC (unknown origin)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Publication
Mercaptoacetamide: A promising zinc-binding group for the discovery of selective histone deacetylase 6 inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 5.30 | 5.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5280773 | — | — | 1 | 5.77 |
| CHEMBL5285554 | — | — | 1 | 5.52 |
| CHEMBL5270758 | — | — | 1 | 4.60 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5280773 | — | IC50 | = | 1700.0 | nM | 5.77 |
| CHEMBL5285554 | — | IC50 | = | 3020.0 | nM | 5.52 |
| CHEMBL5270758 | — | IC50 | = | 25100.0 | nM | 4.60 |