Assay Detail
Binding
CHEMBL5227119
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of PARP1 (unknown origin) using NAD+ as substrate incubated for 60 mins by ELISA
2
Total Activities
1
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Targeting Bromodomain and Extraterminal Proteins for Drug Discovery: From Current Progress to Technological Development.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 5.34 | 5.34 |
| Inhibition | 1 | - | - |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5205994 | — | — | 2 | 5.34 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5205994 | — | IC50 | = | 4600.0 | nM | 5.34 |
| CHEMBL5205994 | — | Inhibition | < | 60.0 | % | - |