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Assay Detail

CHEMBL5227151

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiproliferative activity against human MGC-803 cells assessed as reduction in cell viability incubated for 5 days by MTT assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type MGC-803
Confidence 1 — Organism
Curated By Autocuration

Target

MGC-803 (CHEMBL3706566)
Type CELL-LINE
Organism Homo sapiens

Publication

Reversible Lysine Specific Demethylase 1 (LSD1) Inhibitors: A Promising Wrench to Impair LSD1.
Dai XJ, Liu Y, Xue LP, Xiong XP, Zhou Y, Zheng YC, Liu HM.
J Med Chem (2021) 64 : 2466 -2488
PubMed 33619958 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.06 5.06

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL485818 BAICALIN 1 5.06

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL485818 BAICALIN IC50 = 8780.0 nM 5.06