Assay Detail
Binding
CHEMBL5228230
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Inhibition of RXRbeta (unknown origin)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Targeting Nuclear Receptors in Neurodegeneration and Neuroinflammation.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 3 | 7.57 | 7.64 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5289973 | — | — | 1 | 7.64 |
| CHEMBL114640 | — | — | 1 | 7.62 |
| CHEMBL5279494 | — | — | 1 | 7.44 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5289973 | — | EC50 | = | 23.0 | nM | 7.64 |
| CHEMBL114640 | — | EC50 | = | 24.0 | nM | 7.62 |
| CHEMBL5279494 | — | EC50 | = | 36.0 | nM | 7.44 |