Assay Detail
Binding
CHEMBL5228239
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of Gal4-fused Nur77-LBD in human BGC-823 cells
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | BGC-823 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Nuclear receptor subfamily 4immunitygroup A member 1 (CHEMBL1293229) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Targeting Nuclear Receptors in Neurodegeneration and Neuroinflammation.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1 | 9.94 | 9.94 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1221517 | CYTOSPORONE B | — | 1 | 9.94 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1221517 | CYTOSPORONE B | EC50 | = | 0.115 | nM | 9.94 |