Assay Detail
Binding
CHEMBL5228414
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of aromatase in human JEG-3 cells
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | JEG-3 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Rational Multitargeted Drug Design Strategy from the Perspective of a Medicinal Chemist.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 9.20 | 9.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL108425 | — | — | 1 | 9.30 |
| CHEMBL108483 | — | — | 1 | 9.09 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL108425 | — | IC50 | = | 0.5 | nM | 9.30 |
| CHEMBL108483 | — | IC50 | = | 0.82 | nM | 9.09 |