Assay Detail
Binding
CHEMBL5228419
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Binding affinity to calcium channel alpha2delta1 (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Voltage-dependent calcium channel subunit alpha-2/delta-1 (CHEMBL1919) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Rational Multitargeted Drug Design Strategy from the Perspective of a Medicinal Chemist.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 7.15 | 7.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5273513 | — | — | 1 | 7.96 |
| CHEMBL4745144 | — | — | 1 | 6.34 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5273513 | — | Ki | = | 11.0 | nM | 7.96 |
| CHEMBL4745144 | — | Ki | = | 454.0 | nM | 6.34 |