Assay Detail
Binding
CHEMBL5229090
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of Mycobacterium tuberculosis Zmp1
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mycobacterium tuberculosis |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Novel Antimicrobial 8-Hydroxyquinoline-Based Agents: Current Development, Structure-Activity Relationships, and Perspectives.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 6 | 7.27 | 7.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5265803 | — | — | 1 | 7.96 |
| CHEMBL5279638 | — | — | 1 | 6.94 |
| CHEMBL5278814 | — | — | 1 | 6.91 |
| CHEMBL5276179 | — | — | 1 | - |
| CHEMBL5270776 | — | — | 1 | - |
| CHEMBL1368601 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5265803 | — | IC50 | = | 11.0 | nM | 7.96 |
| CHEMBL5279638 | — | IC50 | = | 115.0 | nM | 6.94 |
| CHEMBL5278814 | — | IC50 | = | 123.0 | nM | 6.91 |
| CHEMBL5276179 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL5270776 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL1368601 | — | IC50 | > | 10000.0 | nM | - |