Assay Detail
Binding
CHEMBL5229280
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human full-length recombinant SENP1
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Recent research and development of inhibitors targeting sentrin-specific protease 1 for the treatment of cancers.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.70 | 5.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2012938 | VIALININ A | — | 1 | 5.80 |
| CHEMBL3236516 | — | — | 1 | 5.60 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2012938 | VIALININ A | IC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL3236516 | — | IC50 | = | 2500.0 | nM | 5.60 |