Assay Detail
Binding
CHEMBL5230787
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Inhibition of HDAC (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Publication
A comprehensive insight on the recent development of Cyclic Dependent Kinase inhibitors as anticancer agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.55 | 5.56 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5280632 | — | — | 1 | 5.56 |
| CHEMBL5280858 | — | — | 1 | 5.53 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5280632 | — | IC50 | = | 2760.0 | nM | 5.56 |
| CHEMBL5280858 | — | IC50 | = | 2950.0 | nM | 5.53 |