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Assay Detail

CHEMBL5230970

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human MDA-MB-231 cells assessed as inhibition of cell growth by MTT assay
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type MDA-MB-231
Confidence 1 — Organism
Curated By Autocuration

Target

MDA-MB-231 (CHEMBL400)
Type CELL-LINE
Organism Homo sapiens

Publication

Hydroxamic acid hybrids as the potential anticancer agents: An Overview.
Liu W, Liang Y, Si X.
Eur J Med Chem (2020) 205 : 112679 -112679
PubMed 32791404 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 6 5.47 6.22

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5287395 1 6.22
CHEMBL5274330 1 6.21
CHEMBL98 VORINOSTAT 4.0 1 5.87
CHEMBL5288573 1 4.83
CHEMBL5269957 1 4.83
CHEMBL5279301 1 4.83

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5287395 IC50 = 600.0 nM 6.22
CHEMBL5274330 IC50 = 620.0 nM 6.21
CHEMBL98 VORINOSTAT IC50 = 1350.0 nM 5.87
CHEMBL5288573 IC50 = 14670.0 nM 4.83
CHEMBL5269957 IC50 = 14670.0 nM 4.83
CHEMBL5279301 IC50 = 14670.0 nM 4.83