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Assay Detail

CHEMBL5230992

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human MCF7 cells assessed as inhibition of cell growth by SRB assay
5
Total Activities
5
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type MCF7
Confidence 1 — Organism
Curated By Autocuration

Target

MCF7 (CHEMBL387)
Type CELL-LINE
Organism Homo sapiens

Publication

Hydroxamic acid hybrids as the potential anticancer agents: An Overview.
Liu W, Liang Y, Si X.
Eur J Med Chem (2020) 205 : 112679 -112679
PubMed 32791404 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 7.39 9.00
GI50 2 - -

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1336 SORAFENIB 4.0 1 9.00
CHEMBL5290567 1 6.80
CHEMBL98 VORINOSTAT 4.0 1 6.37
CHEMBL5274737 1 -
CHEMBL359744 DOXORUBICIN HYDROCHLORIDE 4.0 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1336 SORAFENIB IC50 = 1.0 nM 9.00
CHEMBL5290567 IC50 = 160.0 nM 6.80
CHEMBL98 VORINOSTAT IC50 = 430.0 nM 6.37
CHEMBL5274737 GI50 = 24900.0 nM -
CHEMBL359744 DOXORUBICIN HYDROCHLORIDE GI50 = 50200.0 nM -