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Assay Detail

CHEMBL5231024

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human ASPC1 cells assessed as inhibition of cell growth by MTT assay
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type ASPC1
Confidence 1 — Organism
Curated By Autocuration

Target

ASPC1 (CHEMBL612588)
Type CELL-LINE
Organism Homo sapiens

Publication

Hydroxamic acid hybrids as the potential anticancer agents: An Overview.
Liu W, Liang Y, Si X.
Eur J Med Chem (2020) 205 : 112679 -112679
PubMed 32791404 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 10 6.30 7.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5266413 1 7.30
CHEMBL5283721 1 7.30
CHEMBL3329991 1 6.31
CHEMBL3342181 1 6.06
CHEMBL5268365 1 6.06
CHEMBL5271817 1 6.06
CHEMBL3342182 1 6.06
CHEMBL5272141 1 6.06
CHEMBL98 VORINOSTAT 4.0 1 5.50
CHEMBL5272150 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5266413 IC50 = 50.0 nM 7.30
CHEMBL5283721 IC50 = 50.0 nM 7.30
CHEMBL3329991 IC50 = 490.0 nM 6.31
CHEMBL3342181 IC50 = 880.0 nM 6.06
CHEMBL5268365 IC50 = 880.0 nM 6.06
CHEMBL5271817 IC50 = 880.0 nM 6.06
CHEMBL3342182 IC50 = 880.0 nM 6.06
CHEMBL5272141 IC50 = 880.0 nM 6.06
CHEMBL98 VORINOSTAT IC50 = 3200.0 nM 5.50
CHEMBL5272150 IC50 > 3050.0 nM -