Assay Detail
Binding
CHEMBL5232453
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of BRD9 (unknown origin) by Isothermal titration calorimetry
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
From Hit Seeking to Magic Bullets: The Successful Union of Epigenetic and Fragment Based Drug Discovery (EPIDD + FBDD).
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 3 | 6.61 | 7.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3753082 | — | — | 1 | 7.00 |
| CHEMBL5267719 | — | — | 1 | 6.21 |
| CHEMBL216146 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3753082 | — | Kd | = | 99.0 | nM | 7.00 |
| CHEMBL5267719 | — | Kd | = | 612.0 | nM | 6.21 |
| CHEMBL216146 | — | Kd | = | 5.0 | nM | - |