Assay Detail
Binding
CHEMBL5233293
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inverse agonist activity at human full-length 5-HT2A
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Progress in mechanistically novel treatments for schizophrenia.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 8.73 | 8.73 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2111101 | PIMAVANSERIN | 4.0 | 1 | 8.73 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2111101 | PIMAVANSERIN | IC50 | = | 1.862 | nM | 8.73 |