Assay Detail
Binding
CHEMBL5233329
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human CNT1
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Expanding the repertoire of methanocarba nucleosides from purinergic signaling to diverse targets.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.28 | 4.31 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5270911 | — | — | 1 | 4.31 |
| CHEMBL5285935 | — | — | 1 | 4.24 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5270911 | — | IC50 | = | 49000.0 | nM | 4.31 |
| CHEMBL5285935 | — | IC50 | = | 57000.0 | nM | 4.24 |