Assay Detail
Binding
CHEMBL5234263
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Inhibition of MMP-3 (unknown origin)
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Matrix metalloproteinase-9 (MMP-9) and its inhibitors in cancer: A minireview.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 4 | 7.90 | 8.51 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL437017 | — | — | 1 | 8.51 |
| CHEMBL427616 | — | — | 1 | 8.20 |
| CHEMBL267178 | — | — | 1 | 7.89 |
| CHEMBL34206 | — | — | 1 | 7.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL437017 | — | IC50 | = | 3.1 | nM | 8.51 |
| CHEMBL427616 | — | IC50 | = | 6.3 | nM | 8.20 |
| CHEMBL267178 | — | IC50 | = | 13.0 | nM | 7.89 |
| CHEMBL34206 | — | IC50 | = | 100.0 | nM | 7.00 |