Assay Detail
Binding
CHEMBL5234276
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Inhibition of human MMP2 using Dnp-Pro-Cha-Gly-Cys(Me)-His-Ala-Lys(Nma)-NH2 substrate by fluorimetric analysis
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Matrix metalloproteinase-9 (MMP-9) and its inhibitors in cancer: A minireview.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 9.16 | 9.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL323090 | — | — | 1 | 9.52 |
| CHEMBL5289570 | — | — | 1 | 8.79 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL323090 | — | IC50 | = | 0.3 | nM | 9.52 |
| CHEMBL5289570 | — | IC50 | = | 1.64 | nM | 8.79 |