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Assay Detail

CHEMBL5241503

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiplasmodial activity against Plasmodium falciparum DD2 assessed as growth inhibition
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Plasmodium falciparum
Confidence 1 — Organism
Curated By Autocuration

Target

Plasmodium falciparum (CHEMBL364)
Type ORGANISM
Organism Plasmodium falciparum

Publication

An insight in anti-malarial potential of indole scaffold: A review.
Chauhan M, Saxena A, Saha B.
Eur J Med Chem (2021) 218 : 113400 -113400
PubMed 33823394 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 7.02 7.51

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5286831 1 7.51
CHEMBL5280687 1 7.08
CHEMBL1098875 1 7.00
CHEMBL5269356 1 6.91
CHEMBL5278994 1 6.62

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5286831 IC50 = 31.0 nM 7.51
CHEMBL5280687 IC50 = 84.1 nM 7.08
CHEMBL1098875 IC50 = 100.0 nM 7.00
CHEMBL5269356 IC50 = 123.0 nM 6.91
CHEMBL5278994 IC50 = 238.0 nM 6.62