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Assay Detail

CHEMBL5241642

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiproliferative activity against human ME-180 cells assessed as inhibition of cell growth by [3H]-thymidine incorporation based liquid scintillation counter analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type ME-180
Confidence 1 — Organism
Curated By Autocuration

Target

ME-180 (CHEMBL1075499)
Type CELL-LINE
Organism Homo sapiens

Publication

Overview of all-trans-retinoic acid (ATRA) and its analogues: Structures, activities, and mechanisms in acute promyelocytic leukaemia.
Liang C, Qiao G, Liu Y, Tian L, Hui N, Li J, Ma Y, Li H, Zhao Q, Cao W, Liu H, Ren X.
Eur J Med Chem (2021) 220 : 113451 -113451
PubMed 33895500 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 9.00 9.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL89241 1 9.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL89241 IC50 = 1.0 nM 9.00