Assay Detail
Binding
CHEMBL5242010
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Inhibition of P-selectin (unknown origin) incubated for 30 mins by ELISA
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Non-carbohydrate strategies to inhibit lectin proteins with special emphasis on galectins.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.65 | 6.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5269430 | — | — | 1 | 6.52 |
| CHEMBL293171 | — | — | 1 | 4.77 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5269430 | — | IC50 | = | 300.0 | nM | 6.52 |
| CHEMBL293171 | — | IC50 | = | 17000.0 | nM | 4.77 |