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Assay Detail

CHEMBL5244616

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of DPP4 (unknown origin) using Gly-Pro-7-amido-4-methylcoumarin as substrate incubated for 30 mins by fluorescence analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Dipeptidyl peptidase 4 (CHEMBL284)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Current anti-diabetic agents and their molecular targets: A review.
Kerru N, Singh-Pillay A, Awolade P, Singh P.
Eur J Med Chem (2018) 152 : 436 -488
PubMed 29751237 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 10.05 10.05

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5269668 1 10.05

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5269668 IC50 = 0.09 nM 10.05