Assay Detail
Binding
CHEMBL5246522
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Inhibition of Bacillus licheniformis Proteinase A using Z-GPR-AMC as substrate by fluorescence based analysis
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Bacillus licheniformis |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Ahp-Cyclodepsipeptides as tunable inhibitors of human neutrophil elastase and kallikrein 7: Total synthesis of tutuilamide A, serine protease selectivity profile and comparison with lyngbyastatin 7.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.50 | 7.50 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5284383 | — | — | 1 | 7.50 |
| CHEMBL191881 | LEUPEPTIN | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5284383 | — | IC50 | = | 31.3 | nM | 7.50 |
| CHEMBL191881 | LEUPEPTIN | IC50 | = | 129000.0 | nM | - |