Assay Detail
Binding
CHEMBL5247128
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Inhibition of Acinetobacter baumannii beta-lactamase OXA-235
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Acinetobacter baumannii |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Geminal Diheteroatomic Motifs: Some Applications of Acetals, Ketals, and Their Sulfur and Nitrogen Homologues in Medicinal Chemistry and Drug Design.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.71 | 8.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1257120 | — | — | 1 | 8.10 |
| CHEMBL404 | TAZOBACTAM | 4.0 | 1 | 5.31 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1257120 | — | IC50 | = | 8.0 | nM | 8.10 |
| CHEMBL404 | TAZOBACTAM | IC50 | = | 4880.0 | nM | 5.31 |