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Assay Detail

CHEMBL5253531

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against HCV genotype 1b by replicon assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Hepacivirus hominis
Confidence 1 — Organism
Curated By Autocuration

Target

Hepatitis C virus (CHEMBL379)
Type ORGANISM
Organism Hepacivirus hominis

Publication

2015 Philip S. Portoghese Medicinal Chemistry Lectureship. Curing Hepatitis C Virus Infection with Direct-Acting Antiviral Agents: The Arc of a Medicinal Chemistry Triumph.
Meanwell NA.
J Med Chem (2016) 59 : 7311 -7351
PubMed 27501244 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 6.26 6.26

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL222385 1 6.26

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL222385 EC50 = 550.0 nM 6.26