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Assay Detail

CHEMBL5255494

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against HBV ayw1 infected in human HepG2.2.15 cells
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Hepatitis B virus
Cell Type HepG2.2.15
Confidence 1 — Organism
Curated By Autocuration

Target

Hepatitis B virus (CHEMBL613497)
Type ORGANISM
Organism Hepatitis B virus

Publication

2- and 3-Fluoro-3-deaza-1',6'-isoneplanocin: Synthesis and antiviral properties (including Ebola and Marburg).
Liu C, Chen Q, Schneller SW.
Bioorg Med Chem Lett (2023) 85 : 129219 -129219
PubMed 36898483 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 3 6.65 7.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL141 LAMIVUDINE 4.0 1 7.70
CHEMBL5275097 1 6.37
CHEMBL5279888 1 5.89

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL141 LAMIVUDINE EC50 = 20.0 nM 7.70
CHEMBL5275097 EC50 = 430.0 nM 6.37
CHEMBL5279888 EC50 = 1280.0 nM 5.89