Assay Detail
Binding
CHEMBL5257758
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Antagonist activity at human P2Y6
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Drug-like Antagonists of P2Y Receptors-From Lead Identification to Drug Development.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.22 | 7.43 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1321988 | — | — | 1 | 7.43 |
| CHEMBL5272895 | — | — | 1 | 7.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1321988 | — | IC50 | = | 37.0 | nM | 7.43 |
| CHEMBL5272895 | — | IC50 | = | 100.0 | nM | 7.00 |