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Assay Detail

CHEMBL5259494

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against DENV-2 infected in human Huh-7 cells assessed as reduction in virus-induced cytopathic effect measured after 15 to 30 mins by neutral red based analysis
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism dengue virus type 2
Cell Type Huh-7
Confidence 1 — Organism
Curated By Autocuration

Target

dengue virus type 2 (CHEMBL613966)
Type ORGANISM
Organism dengue virus type 2

Publication

An Isomer of Galidesivir That Potently Inhibits Influenza Viruses and Members of the <i>Bunyavirales</i> Order.
Sparrow KJ, Shrestha R, Wood JM, Clinch K, Hurst BL, Wang H, Gowen BB, Julander JG, Tarbet EB, McSweeney AM, Ward VK, Evans GB, Harris LD.
ACS Med Chem Lett (2023) 14 : 506 -513
PubMed 37077387 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 4 5.73 6.42

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5273609 1 6.42
CHEMBL5276564 1 5.96
CHEMBL1236524 GALIDESIVIR 2.0 1 4.80
CHEMBL5275463 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5273609 EC50 = 380.0 nM 6.42
CHEMBL5276564 EC50 = 1100.0 nM 5.96
CHEMBL1236524 GALIDESIVIR EC50 = 16000.0 nM 4.80
CHEMBL5275463 EC50 > 100000.0 nM -