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Assay Detail

CHEMBL5260669

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Toxicity
Cytotoxicity against human PBMC cells assessed as reduction in cell viability measured after 72 hrs by CellTiter96 Aqueous One Solution cell proliferation assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Toxicity
Organism Homo sapiens
Cell Type PBMC
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Biological evaluation of novel amidino substituted coumarin-benzazole hybrids as promising therapeutic agents.
Beč A, Racané L, Žonja L, Persoons L, Daelemans D, Starčević K, Vianello R, Hranjec M.
RSC Med Chem (2023) 14 : 957 -968
PubMed 37252100 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 5.79 5.80

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5284601 1 5.80
CHEMBL5276739 1 5.77

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5284601 IC50 = 1600.0 nM 5.80
CHEMBL5276739 IC50 = 1700.0 nM 5.77