Assay Detail
Binding
CHEMBL5261123
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Binding affinity to wild type human CXCR2 assessed as dissociation constant
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Structural Analysis of Chemokine Receptor-Ligand Interactions.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 3 | 6.50 | 7.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL38182 | — | — | 1 | 7.00 |
| CHEMBL256668 | — | — | 1 | 6.00 |
| CHEMBL5266300 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL38182 | — | Kd | = | 100.0 | nM | 7.00 |
| CHEMBL256668 | — | Kd | = | 1000.0 | nM | 6.00 |
| CHEMBL5266300 | — | Kd | = | 10000000.0 | nM | - |